|
2008
|
2009
|
2010
|
2011
|
---|
(N = 86)
|
(N = 78)
|
(N = 81)
|
(N = 82)
|
---|
Amodiaquine
|
Median IC50
|
9.6
|
6.5
|
11.2
|
14.5
|
IC50 Range
|
1.6, 1140
|
3.2, 36.7
|
1.0, 45.3
|
2.3, 53.7
|
90th percentile IC50
|
24.0
|
11.8
|
22.2
|
35.4
|
Artemisinin
|
Median IC50
|
3.2
|
8.1
|
9.9
|
10.1
|
IC50 Range
|
1.1, 28.8
|
1.8, 36.7
|
1.9, 38.0
|
1.3, 73.1
|
90th percentile IC50
|
9.3
|
17.0
|
22.4
|
24.9
|
Chloroquine
|
Median IC50
|
30.7
|
15.0
|
22.4
|
76.1
|
IC50 Range
|
1.4, 341.5
|
4.3, 205.5
|
8.1, 430.2
|
4.7, 455.0
|
90th percentile IC50
|
199.4
|
108.2
|
199.1
|
364.6
|
Mefloquine
|
Median IC50
|
34.5
|
44.6
|
32.6
|
41.2
|
IC50 Range
|
1.6, 398.0
|
2.8, 92.1
|
9.2, 75.7
|
1.5, 191.5
|
90th percentile IC50
|
84.6
|
62.5
|
59.0
|
82.4
|
- IC50 values are in nM. IC50 Range = minimum IC50, maximum IC50. 90th percentile IC50 = IC50 value of the 90th percentile within the range of drug responses observed each year.