From: In vitro activity of immunosuppressive drugs against Plasmodium falciparum
Individual IC50and IC90values1 | Median IC50and IC90values | |||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|
3d7 | 7G8 | Dd2 | Strain 1 | Strain 2 | CQr2parasites | |||||||
IC50 | IC90 | IC50 | IC90 | IC50 | IC90 | IC50 | IC90 | IC50 | IC90 | IC50 | IC90 | |
Mycophenolic acid | 5.3 | 15.1 | 5.4 | 15.3 | 5.7 | 16.7 | 5.4 | 14.4 | 6.4 | 23.7 | 5.6 (5.4-5.9)3 | 16 (15.1-18.5) |
Rapamycin | 8.1 | 12.5 | 6.7 | 11.8 | 6.6 | 12.3 | 7.2 | 12.7 | 7.8 | 12.7 | 6.9 (6.6-7.4) | 12.5 (12.2-12.7) |
Everolimus | 7.5 | 11.8 | 5.1 | 10.7 | 6.4 | 11.5 | 5.8 | 11.2 | 6.2 | 11.6 | 6 (5.7-6.3) | 11.3 (11.1-11.5) |
Chloroquine | 0.01 | 0.03 | 0.19 | 1.05 | 0.22 | 1.09 | 0.21 | 0.65 | 0.27 | 0.73 | 0.21 (0.2-0.23) | 0.9 (0.7-1.1) |