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Table 1 Metabolic stability of strasseriolides A–D

From: Preclinical evaluation of strasseriolides AD, potent antiplasmodial macrolides isolated from Strasseria geniculata CF-247,251

 

T1/2

Clint

Clearance

Strasseriolide

(min)

(mL/min/mg)

Category

A

6.47 ± 1.05

103.28 ± 22.6

High

B

8.7 ± 2.4

76.81 ± 9.8

High

C

15.91 ± 1.15

42.00 ± 1.92

Medium

D

>60

>11.13

Low