From: Haematological response in experimental human Plasmodium falciparum and Plasmodium vivax malaria
Pf3D7 (n = 168) Drugs (n) | Nadir, g/L (median, IQR) | Fractional Fall (%, median, IQR) | Day post treatment of Hb Nadir (median, IQR) |
---|---|---|---|
ACT-451840 (1) | 136 | 9.33 | 9 |
DSM265 (12) | 135 (130–141) | 10.9 (10.4–12.9) | 21 (14–23) |
DSM265 + Artefenomel (7) | 115 (114–139) | 10.6 (6.1–11.6) | 21 (20–28) |
Ferroquine (8) | 129 (118–133) | 11.3 (9.3–12.8) | 20 (18–21) |
Griseofulvin (3) | 140 (136–146) | 8.5 (6.8–9.3) | 11 (4–20) |
Cipargamin (4) | 139 (133–144) | 10.0 (8.0–13.0) | 20 (12–23) |
M5717 (20) | 136 (132–142) | 10.6 (8.5–12.9) | 10 (6–14) |
MMV048 (13) | 138 (131–143) | 11.4 (8.4–14.2) | 9 (8–12) |
Mefloquine (22) | 127 (120–139) | 9.1 (7.9–14.7) | 4 (0–9) |
Artefenomel (16) | 125 (119–139) | 8.6 (7.5–9.7) | 8 (1–21) |
Artefenomel + Piperaquine (21) | 132 (127–140) | 9.1 (7.0–13.2) | 14 (0–27) |
Piperaquine (23) | 129 (120–140) | 10.8 (6.3–13.0) | 19 (0–23) |
Piperaquine + Primaquine (2) | 127–138 | 4.2–13.0 | 7–20 |
SJ733 (10) | 136 (130–140) | 9.8 (8.3–11.6) | 12 (10–20) |
ZY-19849 (6) | 128 (122–137) | 10.9 (5.5–11.6) | 7 (3–8) |