Molecule | Chemical structure | Anti- P. falciparum activity (IC50in μM)* | |
---|---|---|---|
W2( CQ- R) | 3D7l( CQ- S) | ||
CQAn28 |
| 0.71 ± 0.03 | 14.87 ± 3.58 |
CQAn33 |
| 0.02 ± 0.001 | 1.17 ± 0.10 |
CQAn34 |
| 0.23 ± 0.15 | 0.3 ± 0.01 |
CQAn37 |
| 0.07 ± 0.03 | 0.57 ± 0.24 |
CQAn39 |
| 0.64 ± 0.29 | 2.39 ± 0.11 |
CQAn45 |
| 0.77 ± 0.21 | 1.17 ± 0.00 |
Chloroquine |
| 0.38±0.03 | 0.081 ± 0.019 |