Bruceantin
|
Eukaryotic (Pf cytoplasmic ribosomes)
|
Inhibits initiation
|
[16, 17]
|
Verrucarin A
|
Eukaryotic (Pf cytoplasmic ribosomes)
|
Inhibits initiation, binds between P- & A- sites
|
[13,14,15]
|
Suramin
|
Eukaryotic (Pf cytoplasmic ribosomes)
|
Inhibits initation & elongation, multiple binding sites
|
[18]
|
Anisomycin
|
Eukaryotic (Pf cytoplasmic ribosomes)
|
Inhibits elongation, binds A-site
|
[13, 17]
|
Cycloheximide
|
Eukaryotic (Pf cytoplasmic ribosomes)
|
Inhibits elongation, binds E-site
|
[13]
|
Homoharringtonine
|
Eukaryotic (Pf cytoplasmic ribosomes)
|
Inhibits elongation on re-initiating ribosomes, binds A-site
|
[13, 20]
|
Lactimidomycin
|
Eukaryotic (Pf cytoplasmic ribosomes)
|
Inhibits elongation, binds E-site
|
[13]
|
Nagilactone C
|
Eukaryotic (Pf cytoplasmic ribosomes)
|
Inhibits elongation, binds A-site
|
[13, 21]
|
Puromycin
|
Pan-inhibitor
|
tRNA mimetic
|
[23, 24]
|
Halofuginone
|
Eukaryotic
|
Inhibits glutamyl-prolyl-tRNA synthetase
|
[22]
|
Thiostrepton
|
Prokaryotic (Pf mitochondrial & apicoplast ribosomes)
|
Inhibits initiation & elongation
|
[25,26,27,28,29,30,– 31]
|